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Identification of selective inhibitors of indoleamine 2,3-dioxygenase 2

Supun M. Bakmiwewa, Amos A. Fatokun, Anh Tran, Richard J. Payne, Nicholas H. Hunt, Helen J. Ball

Bioorganic & Medicinal Chemistry Letters · 2012 · 55 citations · 22 references

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22

Extra Precision Glide:  Docking and Scoring Incorporating a Model of Hydrophobic Enclosure for Protein−Ligand Complexes

Richard A. Friesner, Robert B. Murphy, Matthew P. Repasky et al. · Journal of Medicinal Chemistry · 2006 · 6.9K citations

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Inhibition of indoleamine 2,3-dioxygenase, an immunoregulatory target of the cancer suppression gene Bin1, potentiates cancer chemotherapy

Alexander J. Muller, James B. DuHadaway, Preston S. Donover et al. · Nature Medicine · 2005 · 1.1K citations

, , +16

Inhibition of Indoleamine 2,3-Dioxygenase in Dendritic Cells by Stereoisomers of 1-Methyl-Tryptophan Correlates with Antitumor Responses

De-Yan Hou, Alexander J. Muller, Madhav Sharma et al. · Cancer Research · 2007 · 583 citations

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Reversal of tumoral immune resistance by inhibition of tryptophan 2,3-dioxygenase

Luc Pilotte, Pierre Larrieu, Vincent Stroobant et al. · Proceedings of the National Academy of Sciences · 2012 · 570 citations · Full text

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Novel Tryptophan Catabolic Enzyme IDO2 Is the Preferred Biochemical Target of the Antitumor Indoleamine 2,3-Dioxygenase Inhibitory Compound <scp>d</scp> -1-Methyl-Tryptophan

Richard Metz, James B. DuHadaway, Uma Kamasani et al. · Cancer Research · 2007 · 463 citations · Full text

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