Bioorganic & Medicinal Chemistry · 2004 · 11 citations · 32 references
PharmacyMedicinal ChemistryPharmacologyPharmacodynamicsStructural BiologyStructure-activity RelationshipsLigand BindingMolecular DockingProtein StructureProtein-ligand DockingReceptor-ligand InteractionsStructure-function RelationshipsChemical Structure-activity RelationshipsConformational Changes On BindingConformational MappingStructure-based Binding MechanismsToxin Receptor BindingToxin StructureToxin-receptor Interactions
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The capsaicin receptor: a heat-activated ion channel in the pain pathway
Michael J. Caterina, Mark Schumacher, Makoto Tominaga et al. · Nature · 1997 · 9.1K citations
Impaired Nociception and Pain Sensation in Mice Lacking the Capsaicin Receptor
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The Cloned Capsaicin Receptor Integrates Multiple Pain-Producing Stimuli
Makoto Tominaga, Michael J. Caterina, Annika B. Malmberg et al. · Neuron · 1998 · 3.1K citations · Full text
Vanilloid receptors on sensory nerves mediate the vasodilator action of anandamide
Peter M. Zygmunt, Jesper Petersson, David A. Andersson et al. · Nature · 1999 · 2.1K citations
Vanilloid receptor-1 is essential for inflammatory thermal hyperalgesia
John B. Davis, Julie Gray, Martin J. Gunthorpe et al. · Nature · 2000 · 1.8K citations