Synthesis and biological evaluation of 2-methoxy- and 2-Methylthio-6-[(2′-alkylamino)ethyl]-4(3 H )-pyrimidinones with anti-rubella virus activity

Synthesis and antiviral activity of deoxy analogs of 1-[(2-hydroxyethoxy)methyl]-6-(phenylthio)thymine (HEPT) as potent and selective anti-HIV-1 agents

Hiromichi Tanaka, Hideaki Takashima, Masaru Ubasawa et al. · Journal of Medicinal Chemistry · 1992 · 166 citations

Pharmacy, Medicinal Chemistry, Pharmacology +11

Dihydro(alkylthio)(naphthylmethyl)oxopyrimidines:  Novel Non-Nucleoside Reverse Transcriptase Inhibitors of the <i>S</i>-DABO Series

Antonello Mai, Marino Artico, Gianluca Sbardella et al. · Journal of Medicinal Chemistry · 1997 · 98 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Highly potent and selective inhibition of human immunodeficiency virus type 1 by a novel series of 6-substituted acyclouridine derivatives.

Masanori Baba, Erik De Clercq, H. TANAKA et al. · Molecular Pharmacology · 1991 · 75 citations

Life Sciences, Medicinal Chemistry, Pharmacology +11

Synthesis and Anti-HIV Activity of Novel N-1 Side Chain-Modified Analogs of 1-[(2-Hydroxyethoxy)methyl]-6-(phenylthio)thymine (HEPT)

Renée Pontikis, Rachid Benhida, Anné-Marie Aubertin et al. · Journal of Medicinal Chemistry · 1997 · 72 citations

Pharmacy, Medicinal Chemistry, Pharmacology +16

O-Allyl protection of guanine and thymine residues in oligodeoxyribonucleotides

Yoshihiro Hayakawa, Masaaki Hirose, Ryōji Noyori · The Journal of Organic Chemistry · 1993 · 63 citations

Pharmacy, Molecular Biology, Bioorthogonal Chemistry +9