Concepedia

A bioisosteric approach to the discovery of indole carbinol androgen receptor ligands

James C. Lanter, James J. Fiordeliso, George F. Allan, Amy Musto, Do Won Hahn, Zhihua Sui

Bioorganic & Medicinal Chemistry Letters · 2006 · 19 citations · 6 references

DOIFull text

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Concepts

References

6

Burger's Medicinal Chemistry and Drug Discovery

European Journal of Medicinal Chemistry · 1997 · 681 citations · Full text

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Structural Basis for Accommodation of Nonsteroidal Ligands in the Androgen Receptor

Casey E. Bohl, Duane D. Miller, Jiyun Chen et al. · Journal of Biological Chemistry · 2005 · 209 citations · Full text

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An Efficient Synthesis of 1,2,9,9a-Tetrahydrocyclopropa[c]benz[e]indol-4-one CBI: An Enhanced and Simplified Analog of the CC-1065 and Duocarmycin Alkylation Subunits

Dale L. Boger, Jeffrey A. McKie · The Journal of Organic Chemistry · 1995 · 150 citations

, , +6

Asymmetric hydroformylation of N-acyl 1-aminoacrylic acid derivatives by rhodium/chiral diphosphine catalysts

Serafino Gladiali, Luigi Pinna · Tetrahedron Asymmetry · 1991 · 49 citations

, , +15

Nonsteroidal tissue selective androgen receptor modulators: a promising class of clinical candidates

Michael L. Mohler, Vipin A. Nair, Dong‐Jin Hwang et al. · Expert Opinion on Therapeutic Patents · 2005 · 37 citations

, , +17