Synthesis and antibacterial activity of 3-keto-6-O-carbamoyl-11,12-cyclic thiocarbamate erythromycin A derivatives

Synthesis and antibacterial activity of HMR 3647 a new ketolide highly potent against erythromycin-resistant and susceptible pathogens

Alexis Denis, Constantin Agouridas, Jean-Michel Auger et al. · Bioorganic & Medicinal Chemistry Letters · 1999 · 195 citations

Pharmacy, Medicinal Chemistry, Pharmacology +13

Macrolides, chemistry, pharmacology and clinical uses

H. Vanderhaeghe, Jos Hoogmartens · 1993 · 167 citations

Medicine, Medicinal Chemistry, Pharmacology +12

Novel Erythromycin Derivatives with Aryl Groups Tethered to the C-6 Position Are Potent Protein Synthesis Inhibitors and Active against Multidrug-Resistant Respiratory Pathogens

Zhenkun Ma, Richard F. Clark, Antony Brazzale et al. · Journal of Medicinal Chemistry · 2001 · 112 citations

Pharmacy, Medicinal Chemistry, Pharmacology +17

Recent developments in the area of macrolide antibiotics

Takushi Kaneko, Hamish A. I. McArthur, Joyce A. Sutcliffe · Expert Opinion on Therapeutic Patents · 2000 · 31 citations

Pharmacy, Medicinal Chemistry, Pharmacology +17

Synthesis and antibacterial activity of C2-fluoro, C6-carbamate ketolides, and their C9-oximes

Xiaodong Xu, Todd C. Henninger, Darren Abbanat et al. · Bioorganic & Medicinal Chemistry Letters · 2005 · 25 citations

Natural Sciences, Chemistry, Medicinal Chemistry +8