Constantin Agouridas

Synthesis and Antibacterial Activity of Ketolides (6-<i>O</i>-Methyl-3-oxoerythromycin Derivatives):  A New Class of Antibacterials Highly Potent Against Macrolide-Resistant and -Susceptible Respiratory Pathogens

Constantin Agouridas, Alexis Denis, Jean-Michel Auger et al. · Journal of Medicinal Chemistry · 1998 · 199 citations

Bioorganic Chemistry, Antibacterial Activity, Macrolactone Backbone +21

Synthesis and antibacterial activity of HMR 3647 a new ketolide highly potent against erythromycin-resistant and susceptible pathogens

Alexis Denis, Constantin Agouridas, Jean-Michel Auger et al. · Bioorganic & Medicinal Chemistry Letters · 1999 · 195 citations

Antibiotics, Hmr 3647, Antibacterial Activity +10

The lysine pathway as a target for a new genera of synthetic antibacterial antibiotics?

J.‐M. GIRODEAU, Constantin Agouridas, Maryse Masson et al. · Journal of Medicinal Chemistry · 1986 · 83 citations

Bioorganic Chemistry, Lysine Pathway, Antimicrobial Chemotherapy +24

Antibacterial activity of RU 64004 (HMR 3004), a novel ketolide derivative active against respiratory pathogens

Constantin Agouridas, Alain Bonnefoy, J F Chantot · Antimicrobial Agents and Chemotherapy · 1997 · 57 citations · Full text

Antibacterial Activity, Antimicrobial Chemotherapy, Antibiotic Resistance +16

β-Keto-ester chemistry and ketolides. synthesis and antibacterial activity of 2-halogeno, 2-methyl and 2,3 enol-ether ketolides

Alexis Denis, François Bretin, C Fromentin et al. · Bioorganic & Medicinal Chemistry Letters · 2000 · 52 citations

Halogenation, β-Keto-ester Chemistry, Engineering +7