Concepedia

Synthesis of phenylglycine derivatives as potent and selective antagonists of group III metabotropic glutamate receptors

Stuart J. Conway, Jacqueline C. Miller, Patrick A. Howson, Barry P. Clark, David E. Jane

Bioorganic & Medicinal Chemistry Letters · 2001 · 22 citations · 10 references

DOI

Concepts

References

10

THE EFFECTS OF A SERIES OF ω‐PHOSPHONIC α‐CARBOXYLIC AMINO ACIDS ON ELECTRICALLY EVOKED AND EXCITANT AMINO ACID‐INDUCED RESPONSES IN ISOLATED SPINAL CORD PREPARATIONS

Richard H. Evans, A. A. Francis, Alan Wayne Jones et al. · British Journal of Pharmacology · 1982 · 466 citations · Full text

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Actions of two new antagonists showing selectivity for different sub‐types of metabotropic glutamate receptor in the neonatal rat spinal cord

David E. Jane, Philip L. Jones, P.C‐K. Pook et al. · British Journal of Pharmacology · 1994 · 185 citations · Full text

, , +17

Potent antagonists at the L-AP4- and (1S,3S)-ACPD-sensitive presynaptic metabotropic glutamate receptors in the neonatal rat spinal cord

David E. Jane, Nicola Thomas, H-W. Tse et al. · Neuropharmacology · 1996 · 138 citations

, , +16

New phenylglycine derivatives with potent and selective antagonist activity at presynaptic glutamate receptors in neonatal rat spinal cord

David E. Jane, K. Pittaway, David C. Sunter et al. · Neuropharmacology · 1995 · 105 citations

, , +16

Antagonism of presynaptically mediated depressant responses and cyclic AMP-coupled metabotropic glutamate receptors

Martyn C. Kemp, Peter Roberts‎, Peter C.K. Pook et al. · European Journal of Pharmacology Molecular Pharmacology · 1994 · 95 citations

, , +14