Biochemical Pharmacology · 1991 · 54 citations · 17 references
MedicinePharmacokineticsPharmacologyDrug InteractionsEnzymologyMolecular PharmacologyCytochrome P450 EnzymesCytochrome P450 InteractionsCytochrome P450-mediated MetabolismDrug-metabolizing EnzymesEnzyme InhibitionMetabolism InteractionsCyp450-mediated InteractionsCytochrome P450 Enzyme ActivityCytochrome P450 Enzyme InhibitionCytochrome P450 InhibitionCytochrome P450 Selectivity
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The Determination of Enzyme Dissociation Constants
Hans Lineweaver, Dean Burk · Journal of the American Chemical Society · 1934 · 12.1K citations
The determination of enzyme inhibitor constants
Martin Dixon · Biochemical Journal · 1953 · 4.1K citations · Full text
Substituted benzimidazoles inhibit gastric acid secretion by blocking (H+ + K+) ATPase
E. Fellenius, T. Berglindh, George Sachs et al. · Nature · 1981 · 625 citations
Medicine, Biochemistry, Pharmacology +10