Biochemical Journal · 1974 · 936 citations · 3 references
Life SciencesPharmacologyChemical KineticsEnzyme MechanismEnzymologyCatalytic Reaction KineticsEnzyme AssaysEnzyme InhibitionEnzyme KineticsKinetic ModelingMichaelis-menten KineticsEnzyme Inhibition KineticsEnzyme Kinetic AnalysisEnzyme Kinetic ModelsEnzyme Reaction KineticsInhibition ConstantsInhibition KineticsNoncompetitive InhibitionUncompetitive Inhibition
A new method is described for plotting kinetic results for inhibited enzyme-catalysed reactions. It provides a simple way of determining the inhibition constant, K'(i), of an uncompetitive, mixed or non-competitive inhibitor.
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The determination of enzyme inhibitor constants
Martin Dixon · Biochemical Journal · 1953 · 4.1K citations · Full text
Statistical estimations in enzyme kinetics
GN WILKINSON · Biochemical Journal · 1961 · 3.6K citations · Full text