Concepedia

Functional assay and structure–activity relationships of new third-generation P-glycoprotein inhibitors

Henrik Müller, Ilza Pajeva, Christoph Globisch, Michael Wiese

Bioorganic & Medicinal Chemistry · 2007 · 58 citations · 16 references

DOIFull text

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Concepts

References

16

A surface glycoprotein modulating drug permeability in Chinese hamster ovary cell mutants

R. L. Juliano, Victor Ling · Biochimica et Biophysica Acta (BBA) - Biomembranes · 1976 · 3.3K citations

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Communication between Multiple Drug Binding Sites on P-glycoprotein

Catherine Martin, G. Berridge, Christopher F. Higgins et al. · Molecular Pharmacology · 2000 · 415 citations

, , +16

In vitro and in vivo reversal of P-glycoprotein-mediated multidrug resistance by a novel potent modulator, XR9576.

Prakash Mistry, Alistair Stewart, Wendy Dangerfield et al. · PubMed · 2001 · 350 citations

, , +16

The molecular interaction of the high affinity reversal agent XR9576 with P‐glycoprotein

Catherine Martin, G. Berridge, Prakash Mistry et al. · British Journal of Pharmacology · 1999 · 260 citations · Full text

, , +17

Extraction of Hoechst 33342 from the Cytoplasmic Leaflet of the Plasma Membrane by P‐Glycoprotein

Adam B. Shapiro, Victor Ling · European Journal of Biochemistry · 1997 · 169 citations · Full text

, , +13