Synthesis of novel 2-alkyl triazole-3-alkyl substituted quinoline derivatives and their cytotoxic activity

A Stepwise Huisgen Cycloaddition Process: Copper(I)-Catalyzed Regioselective “Ligation” of Azides and Terminal Alkynes

Vsevolod V. Rostovtsev, Luke G. Green, Valery V. Fokin et al. · Angewandte Chemie International Edition · 2002 · 11.5K citations

Natural Sciences, Chemistry, Catalysis +8

Peptidotriazoles on Solid Phase:  [1,2,3]-Triazoles by Regiospecific Copper(I)-Catalyzed 1,3-Dipolar Cycloadditions of Terminal Alkynes to Azides

Christian W. Tornøe, Caspar Christensen, Morten Meldal · The Journal of Organic Chemistry · 2002 · 8.5K citations

Pharmacy, Medicinal Chemistry, Catalysis +12

1,2,3-Triazole-[2,5-Bis-O-(tert-butyldimethylsilyl)-.beta.-D-ribofuranosyl]-3'-spiro-5''-(4''-amino-1'',2''-oxathiole 2'',2''-dioxide) (TSAO) Analogs: Synthesis and Anti-HIV-1 Activity

Rosa Álvarez, Sonsoles Velázquez, Ana San‐Félix et al. · Journal of Medicinal Chemistry · 1994 · 750 citations

Pharmacy, Medicinal Chemistry, Pharmacology +13

Click Chemistry In Situ: Acetylcholinesterase as a Reaction Vessel for the Selective Assembly of a Femtomolar Inhibitor from an Array of Building Blocks

Warren G. Lewis, Luke G. Green, Flavio Grynszpan et al. · Angewandte Chemie International Edition · 2002 · 740 citations

Life Sciences, Biochemistry, Medicinal Chemistry +16

Synthesis and Antibacterial Evaluation of Certain Quinolone Derivatives

Yeh‐Long Chen, Kuo‐Chang Fang, Shu‐Lin Hsu et al. · Journal of Medicinal Chemistry · 2001 · 550 citations

Pharmacy, Medicinal Chemistry, Pharmacology +12