Correlation between emetic effect of phosphodiesterase 4 inhibitors and their occupation of the high-affinity rolipram binding site in Suncus murinus brain

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

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LIGAND: A versatile computerized approach for characterization of ligand-binding systems

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Deletion of phosphodiesterase 4D in mice shortens α2-adrenoceptor–mediated anesthesia, a behavioral correlate of emesis

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Deletion of phosphodiesterase 4D in mice shortens α2-adrenoceptor–mediated anesthesia, a behavioral correlate of emesis

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Stereospecific binding of the antidepressant rolipram to brain protein structures

Herbert H. Schneider, Ralph Schmiechen, Marina Brezinski et al. · European Journal of Pharmacology · 1986 · 236 citations

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