Concepedia

Structure-based design of novel human Pin1 inhibitors (I)

Chuangxing Guo, Xinjun Hou, Liming Dong, Eleanor Dagostino, S.E. Greasley, Rose Ann Ferre, Joseph Marakovits, M. Catherine Johnson, David A. Matthews, Barbara Mroczkowski,

Bioorganic & Medicinal Chemistry Letters · 2009 · 105 citations · 25 references

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References

25

A human peptidyl–prolyl isomerase essential for regulation of mitosis

Kun Ping Lu, Steven D. Hanes, Tony Hunter · Nature · 1996 · 905 citations

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Structural and Functional Analysis of the Mitotic Rotamase Pin1 Suggests Substrate Recognition Is Phosphorylation Dependent

Rama Ranganathan, Kun Ping Lu, Tony Hunter et al. · Cell · 1997 · 704 citations · Full text

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Function of WW Domains as Phosphoserine- or Phosphothreonine-Binding Modules

Pei‐Jung Lu, Xiao Zhen Zhou, Minhui Shen et al. · Science · 1999 · 684 citations

, , +15

5‐Substituted 1H‐Tetrazoles as Carboxylic Acid Isosteres: Medicinal Chemistry and Synthetic Methods

R. Jason Herr · ChemInform · 2003 · 681 citations

, , +10

Molecular recognition of the inhibitor AG-1343 by HIV-1 protease: conformationally flexible docking by evolutionary programming

Daniel K. Gehlhaar, Gennady M. Verkhivker, Paul A. Rejto et al. · Chemistry & Biology · 1995 · 678 citations · Full text

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