Concepedia

Structure-based design of novel human Pin1 inhibitors (I)

Chuangxing Guo, Xinjun Hou, Liming Dong, Eleanor Dagostino, S.E. Greasley, Rose Ann Ferre, Joseph Marakovits, M. Catherine Johnson, David A. Matthews, Barbara Mroczkowski,

Bioorganic & Medicinal Chemistry Letters · 2009 · 106 citations · 25 references

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References

25

A human peptidyl–prolyl isomerase essential for regulation of mitosis

Kun Ping Lu, Steven D. Hanes, Tony Hunter · Nature · 1996 · 907 citations

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Structural and Functional Analysis of the Mitotic Rotamase Pin1 Suggests Substrate Recognition Is Phosphorylation Dependent

Rama Ranganathan, Kun Ping Lu, Tony Hunter et al. · Cell · 1997 · 707 citations · Full text

, , +8

Function of WW Domains as Phosphoserine- or Phosphothreonine-Binding Modules

Pei‐Jung Lu, Xiao Zhen Zhou, Minhui Shen et al. · Science · 1999 · 686 citations

, , +17

Molecular recognition of the inhibitor AG-1343 by HIV-1 protease: conformationally flexible docking by evolutionary programming

Daniel K. Gehlhaar, Gennady M. Verkhivker, Paul A. Rejto et al. · Chemistry & Biology · 1995 · 685 citations · Full text

, , +17

5‐Substituted 1H‐Tetrazoles as Carboxylic Acid Isosteres: Medicinal Chemistry and Synthetic Methods

R. Jason Herr · ChemInform · 2003 · 681 citations

, , +15