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Nonsteroidal progesterone receptor antagonists based on a conformationally-restricted subseries of 6-aryl-1,2-dihydro-2,2,4-trimethylquinolines

Lawrence G. Hamann, David T. Winn, Charlotte L. F. Pooley, Christopher M. Tegley, Sarah J. West, Luc J. Farmer, James P. Edwards, Keith B. Marschke, Dale E. Mais, Mark E. Goldman,

Bioorganic & Medicinal Chemistry Letters · 1998 · 22 citations · 17 references

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17

2,4-Diamino-5-benzylpyrimidines and analogs as antibacterial agents. 12. 1,2-Dihydroquinolylmethyl analogs with high activity and specificity for bacterial dihydrofolate reductase

Jay V. Johnson, Barbara S. Rauckman, David P. Baccanari et al. · Journal of Medicinal Chemistry · 1989 · 208 citations · Full text

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Mechanism of the Skraup and Doebner-von Miller quinoline syntheses. Cyclization of .alpha.,.beta.-unsaturated N-aryliminium salts via 1,3-diazetidinium ion intermediates

John J. Eisch, Tomasz Dluzniewski · The Journal of Organic Chemistry · 1989 · 99 citations

, , +7

Interaction of glucocorticoid analogues with the human glucocorticoid receptor

Tina S. Berger, Zahra Parandoosh, Bruce W. Perry et al. · The Journal of Steroid Biochemistry and Molecular Biology · 1992 · 77 citations

, , +12

Nonsteroidal progesterone receptor ligands. 1. 3-Aryl-1-benzoyl-1,4,5,6- tetrahydropyridazines.

Donald W. Combs, Kimberly Reese, A. Phillips · Journal of Medicinal Chemistry · 1995 · 73 citations · Full text

, , +9

5-Aryl-1,2-dihydrochromeno[3,4-<i>f</i>]quinolines:  A Novel Class of Nonsteroidal Human Progesterone Receptor Agonists

Lin Zhi, Christopher M. Tegley, E. Adam Kallel et al. · Journal of Medicinal Chemistry · 1998 · 65 citations · Full text

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