SAR-based optimization of 2-(1H-pyrazol-1-yl)-thiazole derivatives as highly potent EP1 receptor antagonists

Masakazu Atobe, Kenji Naganuma, Masashi Kawanishi, Akifumi Morimoto, K. Kasahara, Shigeki Ohashi, Hiroko Suzuki, Takahiko Hayashi, Shiro Miyoshi

Bioorganic & Medicinal Chemistry Letters · 2013 · 18 citations · 9 references

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