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Synthesis and Biological Evaluation of the 1,5-Diarylpyrazole Class of Cyclooxygenase-2 Inhibitors:  Identification of 4-[5-(4-Methylphenyl)-3- (trifluoromethyl)-1<i>H</i>-pyrazol-1-yl]benzenesulfonamide (SC-58635, Celecoxib)

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NS-398, a new anti-inflammatory agent, selectively inhibits prostaglandin G/H synthase/cyclooxygenase (COX-2) activity in vitro

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Detection and Isolation of an Endoperoxide Intermediate in Prostaglandin Biosynthesis

Mats Hámberg, Bengt Samuelsson · Proceedings of the National Academy of Sciences · 1973 · 644 citations · Full text

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