Concepedia

Solvent free synthesis of 1,5-disubstituted tetrazoles derived from Baylis Hillman acetates as potential TNF-α inhibitors

Palash Dutta, R. Srinivasa Rao, J. S. Yadav, S. Chandrasekhar, Pravin Thombare, Jogeswar Mohapatra, Abhijit Chatterjee, Mukul R. Jain

Bioorganic & Medicinal Chemistry Letters · 2009 · 55 citations · 21 references

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References

21

Preparation of 5-Substituted 1<i>H</i>-Tetrazoles from Nitriles in Water

Zachary Demko, K. Barry Sharpless · The Journal of Organic Chemistry · 2001 · 962 citations

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5-Substituted-1H-tetrazoles as carboxylic acid isosteres: medicinal chemistry and synthetic methods

R. Jason Herr · Bioorganic & Medicinal Chemistry · 2002 · 844 citations

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5‐Substituted 1H‐Tetrazoles as Carboxylic Acid Isosteres: Medicinal Chemistry and Synthetic Methods

R. Jason Herr · ChemInform · 2003 · 681 citations

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A click chemistry approach to tetrazoles by Huisgen 1,3-dipolar cycloaddition: synthesis of 5-acyltetrazoles from azides and acyl cyanides.

Zachary Demko, K. Barry Sharpless · PubMed · 2002 · 447 citations

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Nonpeptide angiotensin II receptor antagonists: the discovery of a series of N-(biphenylylmethyl)imidazoles as potent, orally active antihypertensives

David J. Carini, John V. Duncia, Paul E. Aldrich et al. · Journal of Medicinal Chemistry · 1991 · 431 citations · Full text

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