5-Substituted-1H-tetrazoles as carboxylic acid isosteres: medicinal chemistry and synthetic methods

Methods for drug discovery: development of potent, selective, orally effective cholecystokinin antagonists

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Preparation of 5-Substituted 1<i>H</i>-Tetrazoles from Nitriles in Water

Zachary Demko, K. Barry Sharpless · The Journal of Organic Chemistry · 2001 · 962 citations

Natural Sciences, Chemistry, Catalysis +6

Structure of the HIV-1 integrase catalytic domain complexed with an inhibitor: A platform for antiviral drug design

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Nonpeptide angiotensin II receptor antagonists: the discovery of a series of N-(biphenylylmethyl)imidazoles as potent, orally active antihypertensives

David J. Carini, John V. Duncia, Paul E. Aldrich et al. · Journal of Medicinal Chemistry · 1991 · 431 citations · Full text

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An Improved Synthesis of 5-Substituted Tetrazoles

William Finnegan, Ronald A. Henry, Robert Alden Lofquist · Journal of the American Chemical Society · 1958 · 406 citations

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