Concepedia

Estrone and estradiol C-16 derivatives as inhibitors of type 1 17β-hydroxysteroid dehydrogenase

Donald Poirier, Ho-Jin Chang, Arezki Azzi, Roch P. Boivin, Sheng‐Xiang Lin

Molecular and Cellular Endocrinology · 2005 · 28 citations · 8 references

DOI

Concepts

References

8

Development and validation of a genetic algorithm for flexible docking 1 1Edited by F. E. Cohen

Gareth Jones, Peter Willett, Robert C. Glen et al. · Journal of Molecular Biology · 1997 · 6.7K citations

, , +14

A concerted, rational design of type 1 17β‐hydroxysteroid dehydrogenase inhibitors: estradiol‐adenosine hybrids with high affinity

Wei Qiu, Robert L. Campbell, Anne Gangloff et al. · The FASEB Journal · 2002 · 85 citations · Full text

, , +17

Overview of a rational approach to design type I 17β-hydroxysteroid dehydrogenase inhibitors without estrogenic activity: chemical synthesis and biological evaluation

Martin Tremblay, Donald Poirier · The Journal of Steroid Biochemistry and Molecular Biology · 1998 · 74 citations

, , +12

17 -Hydroxysteroid dehydrogenase: inhibitors and inhibitor design

T.M. Penning · Endocrine Related Cancer · 1996 · 74 citations

, , +11

Inhibitors of steroidogenesis as agents for the treatment of hormone-dependent cancers

H J Smith, Paul J. Nicholls, Claire Simons et al. · Expert Opinion on Therapeutic Patents · 2001 · 69 citations

, , +17