Replacement of imidazole by a piperidine moiety differentially affects the potency of histamine H3-receptor antagonists

Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

Jean‐Michel Arrang, M. Garbarg, Jean‐Charles Schwartz · Nature · 1983 · 1.6K citations

Brain Histamine Release, Neurophysiology, Medicine +13

Highly potent and selective ligands for histamine H3-receptors

J.M. Arrang, M. Garbarg, J.-C. Lancelo et al. · Nature · 1987 · 900 citations

Biochemistry, Functional Selectivity, Medicine +5

Cloning and Functional Expression of the Human Histamine H₃Receptor

Timothy W. Lovenberg, Barbara Roland, Sandy J. Wilson et al. · Molecular Pharmacology · 1999 · 700 citations · Full text

High constitutive activity of native H3 receptors regulates histamine neurons in brain

Séverine Morisset‐Lopez, A. Rouleau, Xavier Ligneau et al. · Nature · 2000 · 462 citations

Histamine Neurons, Neurophysiology, Synaptic Transmission +12

Pharmacological analysis of drug-receptor interaction

Manfred Kietzmann · Toxicon · 1994 · 225 citations

Drug Interactions, Molecular Pharmacology, Drug Target +5