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Benzoxazole piperidines as selective and potent somatostatin receptor subtype 5 antagonists

Rainer E. Martin, Peter J. Mohr, Hans Peter Maerki, Wolfgang Guba, Christoph Kuratli, Olivier Gavelle, Alfred Binggeli, Stefanie Bendels, Rubén Alvarez‐Sánchez, André Alker,

Bioorganic & Medicinal Chemistry Letters · 2009 · 16 citations · 13 references

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13

Hypothalamic Polypeptide That Inhibits the Secretion of Immunoreactive Pituitary Growth Hormone

Paul Brazeau, Wylie Vale, Roger Burgus et al. · Science · 1973 · 3.5K citations

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Physicochemical High Throughput Screening:  Parallel Artificial Membrane Permeation Assay in the Description of Passive Absorption Processes

Manfred Kansy, Frank Senner, Klaus Gubernator · Journal of Medicinal Chemistry · 1998 · 1.3K citations

, , +16

Subtype-selective expression of the five somatostatin receptors (hSSTR1-5) in human pancreatic islet cells: a quantitative double-label immunohistochemical analysis.

Ujendra Kumar, Ramakrishnan Sasi, Sundar Suresh et al. · Diabetes · 1999 · 286 citations

, , +15

A quantitative assessment of hERG liability as a function of lipophilicity

Michael J. Waring, Craig Johnstone · Bioorganic & Medicinal Chemistry Letters · 2006 · 148 citations

, , +7

Somatostatin-28 regulates GLP-1 secretion via somatostatin receptor subtype 5 in rat intestinal cultures

Connie Chisholm, Gordon R. Greenberg · American Journal of Physiology-Endocrinology and Metabolism · 2002 · 97 citations

, , +17