Concepedia

Estimation of agonist affinity and efficacy by direct, operational model-fitting

P. Leff, D.J. Prentice, Heather Giles, Graeme R. Martin, John N. Wood

Journal of Pharmacological Methods · 1990 · 91 citations · 10 references

DOI

Concepts

References

10

A MODIFICATION OF RECEPTOR THEORY

R. P. STEPHENSON · British Journal of Pharmacology and Chemotherapy · 1956 · 1.1K citations · Full text

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Operational models of pharmacological agonism

J.W. Black, P. Leff · Proceedings of the Royal Society of London. Series B, Biological sciences · 1983 · 1.1K citations

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An operational model of pharmacological agonism: the effect of E/[A] curve shape on agonist dissociation constant estimation

J.W. Black, P. Leff, Nigel P. Shankley et al. · British Journal of Pharmacology · 1985 · 294 citations · Full text

, , +9

Perspectives in receptor classification

Keith Burdett · FEBS Letters · 1988 · 95 citations · Full text

, , +6

?-Adrenoceptor blocking agents as partial agonists in isolated heart muscle: Dissociation of stimulation and blockade

Alberto J. Kaumann, John R. Blinks · Naunyn-Schmiedeberg s Archives of Pharmacology · 1980 · 89 citations

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