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BIOLOGICAL ACTIVITY OF AMINOPHOSPHONIC ACIDS

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Life Sciences, Biochemistry, Pharmacology +11

New hybrid transition state analog inhibitors of HIV protease with peripheric C2-symmetry

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Life Sciences, Medicinal Chemistry, Molecular Biology +13

Preparation of peptidic α-hydroxy phosphonates a new class of transition state analog renin inhibitors

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Pharmacy, Medicinal Chemistry, Pharmacology +12

Asymmetric Hydrogenation of .beta.-Keto Phosphonates: A Practical Way to Fosfomycin

Masato Kitamura, Makoto Tokunaga, Ryōji Noyori · Journal of the American Chemical Society · 1995 · 204 citations

Pharmacy, Biochemistry, Medicinal Chemistry +8

EPSP Synthase: The Design and Synthesis of Bisubstrate Inhibitors Incorporating Novel 3-Phosphate Mimics

James A. Sikorski, Michael J. Miller, Diane S. Braccolino et al. · Phosphorus, sulfur, and silicon and the related elements · 1993 · 130 citations

Life Sciences, Biochemistry, Biocatalysis +12