Concepedia

Design and discovery of 1,3-benzodiazepines as novel dopamine antagonists

Zhaoning Zhu, Z. J. Sun, Yuanzan Ye, Brian A. McKittrick, William J. Greenlee, Michael Czarniecki, Ahmad Fawzi, Hongtao Zhang, Jean E. Lachowicz

Bioorganic & Medicinal Chemistry Letters · 2009 · 27 citations · 16 references

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16

New N- and O-arylations with phenylboronic acids and cupric acetate

Dominic M. T. Chan, Kevin L. Monaco, Ru-Ping Wang et al. · Tetrahedron Letters · 1998 · 1.1K citations

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SCH 23390, a potential benzazepine antipsychotic with unique interactions on dopaminergic systems.

Louis C. Iorio, A Barnett, Frederick H. Leitz et al. · Journal of Pharmacology and Experimental Therapeutics · 1983 · 897 citations

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Effects of ecopipam, a selective dopamine D1 antagonist, on smoked cocaine self-administration by humans

Margaret Haney, Amie S. Ward, Richard W. Foltin et al. · Psychopharmacology · 2001 · 186 citations

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Solid supported CN cross-coupling reactions

Andrew P. Combs, Simon Saubern, Maria Rafalski et al. · Tetrahedron Letters · 1999 · 133 citations

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Dopamine D<sub>1</sub>/D<sub>5</sub> Receptor Antagonists with Improved Pharmacokinetics:  Design, Synthesis, and Biological Evaluation of Phenol Bioisosteric Analogues of Benzazepine D<sub>1</sub>/D<sub>5</sub> Antagonists

Wen‐Lian Wu, Duane A. Burnett, Richard Spring et al. · Journal of Medicinal Chemistry · 2005 · 93 citations

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