Concepedia

Synthesis and anti-HIV activity of 2-naphthyl substituted DAPY analogues as non-nucleoside reverse transcriptase inhibitors

Yonghong Liang, Qiuqin He, Zhao‐Sen Zeng, Zhi‐Qian Liu, Xiaoqing Feng, Fen‐Er Chen, Jan Balzarini, Christophe Pannecouque, Erik De Clercq

Bioorganic & Medicinal Chemistry · 2010 · 37 citations · 9 references

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References

9

Rapid and automated tetrazolium-based colorimetric assay for the detection of anti-HIV compounds

Rudi Pauwels, Jan Balzarini, Masanori Baba et al. · Journal of Virological Methods · 1988 · 1.6K citations

, , +12

Tetrazolium-based colorimetric assay for the detection of HIV replication inhibitors: revisited 20 years later

Christophe Pannecouque, Dirk Daelemans, Erik De Clercq · Nature Protocols · 2008 · 349 citations

, , +14

Evolution of anti-HIV drug candidates. Part 3: diarylpyrimidine (DAPY) analogues

Donald Ludovici, Bart L. De Corte, Michael J. Kukla et al. · Bioorganic & Medicinal Chemistry Letters · 2001 · 185 citations

, , +12

Synthesis of Novel Diarylpyrimidine Analogues and Their Antiviral Activity against Human Immunodeficiency Virus Type 1

Jérôme Guillemont, Élisabeth Pasquier, Patrice Palandjian et al. · Journal of Medicinal Chemistry · 2004 · 118 citations

, , +16

Synthesis of novel diarylpyrimidine analogues of TMC278 and their antiviral activity against HIV-1 wild-type and mutant strains

Céline Mordant, Benoît Schmitt, Élisabeth Pasquier et al. · European Journal of Medicinal Chemistry · 2006 · 70 citations

, , +16