Concepedia
Tetrahedron Letters · 2000 · 27 citations · 4 references
MedicineMechanism Of ActionPharmacological AgentPharmacotherapyPharmacologyDrug Discovery
4
Efficient Synthesis of Losartan, A Nonpeptide Angiotensin II Receptor Antagonist
Robert D. Larsen, Anthony O. King, Cheng‐Yu Chen et al. · The Journal of Organic Chemistry · 1994 · 191 citations
Cardiovascular Pharmacology, Altmetric Attention Score, Peptide Science +17
Nonpeptide angiotensin II receptor antagonists. Synthesis and biological activity of benzimidazolecarboxylic acids
Keiji Kubo, Yasuhisa Kohara, Eiko Imamiya et al. · Journal of Medicinal Chemistry · 1993 · 135 citations · Full text
Biological Activity, Molecular Pharmacology, Medicinal Chemistry +15
Tetrakis(dimethylamino)ethylene as a Useful Reductant of Some Bromodifluoromethyl Heterocycles. Application to the Synthesis of New <i>gem</i>-Difluorinated Heteroarylated Compounds
Conrad R. Burkholder, William R. Dolbier, Maurice Médebielle · The Journal of Organic Chemistry · 1998 · 103 citations
New nonpeptide angiotensin II receptor antagonists. 1. Synthesis, biological properties and structure-activity relationships of 2-alkylbenzimidazole derivatives
Andrew P. Thomas, C. Allott, Keith H. Gibson et al. · Journal of Medicinal Chemistry · 1992 · 91 citations · Full text