Solution-phase combinatorial synthesis of isoxazolines and isoxazoles using [2+3] cycloaddition reaction of nitrile oxides

Drug Discovery: A Historical Perspective

Jürgen Drews · Science · 2000 · 2.7K citations

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Combinatorial Materials Science and Catalysis

Bernd Jandeleit, D. Schaefer, Timothy S. Powers et al. · Angewandte Chemie International Edition · 1999 · 616 citations

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Ti-Catalyzed Regio- and Enantioselective Synthesis of Unsaturated α-Amino Nitriles, Amides, and Acids. Catalyst Identification through Screening of Parallel Libraries

James Porter, Wolfgang Wirschun, Kevin W. Kuntz et al. · Journal of the American Chemical Society · 2000 · 113 citations

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A strategic alternative to solid phase synthesis: Preparation of a small isoxazoline library by “fluorous synthesis”

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Pharmacy, Chemistry, Medicinal Chemistry +12

β-Cyclodextrin as a Scaffold for Supramolecular Chemistry, To Reverse the Regioselectivity of Nitrile Oxide Cycloadditions

Adam G. Meyer, Christopher J. Easton, Stephen F. Lincoln et al. · The Journal of Organic Chemistry · 1998 · 23 citations

Natural Sciences, Chemistry, Medicinal Chemistry +16