Concepedia

Synthesis of 3-Nitrosoimidazo[1,2-a]pyridine Derivatives as Potential Antiretroviral Agents

Aziz Chaouni-Benabdallah, Christophe Galtier, H. Allouchi, Abdelhak Kherbeche, Jean‐Claude Debouzy, Jean-Claude Teulade, Olivier Chavignon, Myriam Witvrouw, Christophe Pannecouque, Jan Balzarini,

Archiv der Pharmazie · 2001 · 20 citations · 15 references

DOI

Concepts

Abstract

Ten 2-aryl or heteroaryl-3-nitrosoimidazo[1,2-a]pyridine derivatives were synthesised as potential antiretroviral agents. The new compounds were characterized by elemental analysis, 1H NMR, and by crystallography for (14). The compounds were devoid of any activity against HIV-1 or HIV-2.

References

15

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Synthesis of Acyclo-<i>C</i>-nucleosides in the Imidazo[1,2-<i>a</i>]pyridine and Pyrimidine Series as Antiviral Agents

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