Synthesis of new pyridazino[4,5-b]indol-4-ones and pyridazin-3(2H)-one analogs as DYRK1A inhibitors

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Development of a novel selective inhibitor of the Down syndrome-related kinase Dyrk1A

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β-Carboline Compounds, Including Harmine, Inhibit DYRK1A and Tau Phosphorylation at Multiple Alzheimer's Disease-Related Sites

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DNA binding properties of 9-substituted harmine derivatives

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Natural Sciences, 9-Substituted Harmine Derivatives, Molecular Biology +4

Structures of Down Syndrome Kinases, DYRKs, Reveal Mechanisms of Kinase Activation and Substrate Recognition

M. Soundararajan, A.K. Roos, P. Savitsky et al. · Structure · 2013 · 154 citations · Full text