Bioorganic & Medicinal Chemistry Letters · 1998 · 18 citations · 11 references
PharmacyChemistryMedicinal ChemistryDrug DesignOrganic ChemistrySynthetic Medicinal ChemistryEnzyme InhibitionOrganic SynthesisPolymerase Chain ReactionPotency OptimizationEnzyme Inhibitor DiscoveryEnzyme Inhibitor SynthesisNon-nucleoside InhibitorsNon-nucleoside Reverse Transcriptase InhibitorsNonnucleoside InhibitorsTherapeutic Index DeterminationTranscription Inhibitors
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Potent and selective inhibition of HIV-1 replication in vitro by a novel series of TIBO derivatives
Rudi Pauwels, Koen Andries, Jan Desmyter et al. · Nature · 1990 · 757 citations