The first organometallic antioestrogens and their antiproliferative effects

Cloning of a novel receptor expressed in rat prostate and ovary.

George G. J. M. Kuiper, Eva Enmark, Markku Pelto‐Huikko et al. · Proceedings of the National Academy of Sciences · 1996 · 4.8K citations

Life Sciences, Endocrinology, Molecular Biology +12

Molecular basis of agonism and antagonism in the oestrogen receptor

A.M. Brzozowski, A.C.W. Pike, Zbigniew Dauter et al. · Nature · 1997 · 3.3K citations

Life Sciences, Endocrinology, Pharmacology +14

Evaluation of the antitumour activity of the non-steroidal antioestrogen monohydroxytamoxifen in the DMBA-induced rat mammary carcinoma model

V. Craig Jordan, Karen E. Allen · European Journal of Cancer (1965) · 1980 · 214 citations

Medicine, Oncology, Pharmacology +14

Structure−Activity Relationships of Selective Estrogen Receptor Modulators:  Modifications to the 2-Arylbenzothiophene Core of Raloxifene

Timothy A. Grese, Stephen Cho, Don R. Finley et al. · Journal of Medicinal Chemistry · 1997 · 176 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +12

Rhenium Carbonyl Complexes of .beta.-Estradiol Derivatives with High Affinity for the Estradiol Receptor: An Approach to Selective Organometallic Radiopharmaceuticals

Siden Top, Hassane El Hafa, Anne Vessières et al. · Journal of the American Chemical Society · 1995 · 169 citations

Medicine, Chemistry, Pharmacology +10