Biochemical Pharmacology · 1993 · 20 citations · 75 references
PharmacyBiochemistryMolecular BiologyDrug DesignDrug DiscoveryEnzymologyEnzyme InhibitionEnzyme ScreeningHigh-throughput ScreeningMolecular ScreeningSmall-molecule ScreeningVirtual ScreeningInhibitor ScreeningKinase InhibitorsKinase Selectivity ProfilingKinase Substrate SpecificityProtein Kinase Inhibitors
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Genistein, a specific inhibitor of tyrosine-specific protein kinases.
Tetsu Akiyama, Junko Ishida, Shizue Nakagawa et al. · Journal of Biological Chemistry · 1987 · 3.7K citations · Full text
Blocking of EGF-Dependent Cell Proliferation by EGF Receptor Kinase Inhibitors
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Inhibitory effects of the tyrosine kinase inhibitor genistein on mammalian DNA topoisomerase II.
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