Concepedia
Trends in Pharmacological Sciences · 1992 · 754 citations · 24 references
PharmacyMolecular BiologyMolecular RecognitionActive Site ArchitectureBinding AffinityBinding SpecificityRecognition MotifsBinding Site SpecificitySigma Factor InteractionsSigma Factor Recognition
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Evidence for sigma opioid receptor: binding of [3H]SKF-10047 to etorphine-inaccessible sites in guinea-pig brain.
Tsung‐Ping Su · Journal of Pharmacology and Experimental Therapeutics · 1982 · 434 citations
Medicine, Neurobiology, Pharmacology +17
Autoradiographic localization of sigma receptor binding sites in guinea pig and rat central nervous system with (+)3H-3-(3-hydroxyphenyl)-N-(1- propyl)piperidine
AL Gundlach, BL Largent, SH Snyder · Journal of Neuroscience · 1986 · 393 citations · Full text
Medicine, Neuroscience, Pharmacology +14
A sigma-like binding site in rat pheochromocytoma (PC12) cells: decreased affinity for (+)-benzomorphans and lower molecular weight suggest a different sigma receptor form from that of guinea pig brain
Susan B. Hellewell, W. Don Bowen · Brain Research · 1990 · 388 citations
Medicine, Neuroscience, Pharmacology +8
Autoradiographic visualization of haloperidol-sensitive sigma receptors in guinea-pig brain
Stafford McLean, E Weber · Neuroscience · 1988 · 177 citations
Medicine, Neuroscience, Pharmacology +7
Metabolites of haloperidol display preferential activity at σ receptors compared to dopamine D-2 receptors
W. Don Bowen, Eydie L. Moses, Paul J. Tolentino et al. · European Journal of Pharmacology · 1990 · 154 citations
Medicine, Medicinal Chemistry, Pharmacology +15