Concepedia

7-Amino-2-phenylpyrazolo[4,3-d]pyrimidine derivatives: Structural investigations at the 5-position to target human A1 and A2A adenosine receptors. Molecular modeling and pharmacological studies

Lucia Squarcialupi, Vittoria Colotta, Daniela Catarzi, Flavia Varano, Marco Betti, Katia Varani, Fabrizio Vincenzi, Pier Andrea Borea, Nicola Porta, Antonella Ciancetta,

European Journal of Medicinal Chemistry · 2014 · 24 citations · 45 references

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References

45

A Rapid and Sensitive Method for the Quantitation of Microgram Quantities of Protein Utilizing the Principle of Protein-Dye Binding

Mark A. Bradford · Analytical Biochemistry · 1976 · 225.4K citations

, , +7

A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding

Marion M. Bradford · Analytical Biochemistry · 1976 · 211.2K citations

, , +7

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

, , +14

LIGAND: A versatile computerized approach for characterization of ligand-binding systems

Peter J. Munson, David Rodbard · Analytical Biochemistry · 1980 · 8.5K citations

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Structural Basis for Allosteric Regulation of GPCRs by Sodium Ions

Wei Liu, Eugene Chun, Aaron A. Thompson et al. · Science · 2012 · 965 citations · Full text

, , +17