Concepedia

3-(2-Aminocarbonylphenyl)propanoic acid analogs as potent and selective EP3 receptor antagonists. Part 1: Discovery and exploration of the carboxyamide side chain

Masaki Asada, Tetsuo Obitsu, Toshihiko Nagase, Motoyuki Tanaka, Yoshiyuki Yamaura, Hiroya Takizawa, Ken Yoshikawa, Kazutoyo Sato, Masami Narita, Shuichi Ohuchida,

Bioorganic & Medicinal Chemistry · 2009 · 15 citations · 20 references

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References

20

Prostaglandin D2 Selectively Induces Chemotaxis in T Helper Type 2 Cells, Eosinophils, and Basophils via Seven-Transmembrane Receptor Crth2

Hiroyuki Hirai, Kazuya Tanaka, Osamu Yoshie et al. · The Journal of Experimental Medicine · 2001 · 1.1K citations · Full text

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Impaired febrile response in mice lacking the prostaglandin E receptor subtype EP3

Fumitaka Ushikubi, Eri Segi‐Nishida, Yukihiko Sugimoto et al. · Nature · 1998 · 687 citations

, , +12

Characterization of EP receptor subtypes responsible for prostaglandin E<sub>2</sub>‐induced pain responses by use of EP<sub>1</sub> and EP<sub>3</sub> receptor knockout mice

Toshiaki Minami, Hiroyuki Nakano, Takuya Kobayashi et al. · British Journal of Pharmacology · 2001 · 181 citations · Full text

, , +17

Vascular wall–produced prostaglandin E2 exacerbates arterial thrombosis and atherothrombosis through platelet EP3 receptors

Sabrina Gross, Peggy Tilly, Didier Hentsch et al. · The Journal of Experimental Medicine · 2007 · 178 citations · Full text

, , +17

Prostanoid inhibition of canine parietal cells: Mediation by the inhibitory guanosine triphosphate-binding protein of adenylate cyclase

Monica C.Y. Chen, Deborah A. Amirian, Mary Toomey et al. · Gastroenterology · 1988 · 126 citations

, , +13