Evidence for antagonist activity of the dopamine D3 receptor partial agonist, BP 897, at human dopamine D3 receptor

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

Life Sciences, Biochemistry, Chemical Kinetics +14

SOME QUANTITATIVE USES OF DRUG ANTAGONISTS

O. ARUNLAKSHANA, H. O. Schild · British Journal of Pharmacology and Chemotherapy · 1959 · 4K citations · Full text

Medicine, Pharmacology, General Pharmacology +16

Molecular cloning and characterization of a novel dopamine receptor (D3) as a target for neuroleptics

Pierre Sokoloff, Bruno Giros, Marie‐Pascale Martres et al. · Nature · 1990 · 2.6K citations · Full text

Life Sciences, Neuroscience, Pharmacology +12

Selective inhibition of cocaine-seeking behaviour by a partial dopamine D3 receptor agonist

Maria Pilla, Sylvie Perachon, François Sautel et al. · Nature · 1999 · 568 citations

Medicine, Neuroscience, Pharmacology +13

Modulation of Cocaine Self-Administration in the Rat Through D-3 Dopamine Receptors

S. Barak Caine, George F. Koob · Science · 1993 · 455 citations

Medicine, Neuroscience, Pharmacology +12