Concepedia

Efficient and Diverse Synthesis of Indole Derivatives

Haixia Liu, Alexander Dömlingꝉ

The Journal of Organic Chemistry · 2009 · 89 citations · 22 references

DOI

Concepts

Abstract

A convergent 2-step procedure toward an array of indole derivatives involving an Ugi reaction and a Pictet-Spengler reaction is described. The reactions are versatile regarding different starting materials. Hexacyclic 24 can be produced with unprecedented complexity.

References

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