Concepedia

Synthesis and pharmacology of isoquinuclidine derivatives as 5-HT3 ligands

Isabel Iriepa, F. Javier Villasante, Enrique J. Galvez, Luis Labeaga, Ana Innerárity, Aurelio Orjales

Bioorganic & Medicinal Chemistry Letters · 2002 · 21 citations · 10 references

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References

10

A practical computer-based approach to the analysis of radioligand binding experiments

Grant A. McPherson · Computer Programs in Biomedicine · 1983 · 832 citations

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Specific in vitro and in vivo binding of 3H-raclopride a potent substituted benzamide drug with high affinity for dopamine D-2 receptors in the rat brain

Christer Köhler, Håkan Hall, Sven Ove Ögren et al. · Biochemical Pharmacology · 1985 · 506 citations

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Development of a radioligand binding assay for 5‐HT<sub>4</sub> receptors in guinea‐pig and rat brain

Carol J. Grossman, Gavin J. Kilpatrick, K T Bunce · British Journal of Pharmacology · 1993 · 283 citations · Full text

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Novel 5-HT3 antagonists. Indole oxadiazoles

Christopher J. Swain, Robert J. Baker, Clare O. Kneen et al. · Journal of Medicinal Chemistry · 1991 · 167 citations · Full text

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5-Hydroxytryptamine (5-HT3) receptor antagonists. 1. Indazole and indolizine-3-carboxylic acid derivatives

José Luis Bermúdez, Charles S. Fake, Graham F. Joiner et al. · Journal of Medicinal Chemistry · 1990 · 153 citations · Full text

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