Concepedia

Novel Selective Quinazoline Inhibitors of Endothelin Converting Enzyme-1

Kyunghye Ahn, Andre M. Sisneros, Sarah B. Herman, Sharon Pan, Donald Hupe, Chitase Lee, Sham S. Nikam, Xue-Min Cheng, Annette M. Doherty, Richard L. Schroeder,

Biochemical and Biophysical Research Communications · 1998 · 45 citations · 38 references

DOI

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38

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

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A novel potent vasoconstrictor peptide produced by vascular endothelial cells

Masashi Yanagisawa, Hiroki Kurihara, Sadao Kimura et al. · Nature · 1988 · 10.8K citations · Full text

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The human endothelin family: three structurally and pharmacologically distinct isopeptides predicted by three separate genes.

Akiko Inoue, Masashi Yanagisawa, Sadao Kimura et al. · Proceedings of the National Academy of Sciences · 1989 · 2.5K citations · Full text

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Elevated blood pressure and craniofaclal abnormalities in mice deficient in endothelin-1

Yukiko Kurihara, Hiroki Kurihara, Hiroshi Suzuki et al. · Nature · 1994 · 992 citations

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Interaction of endothelin-3 with endothelin-B receptor is essential for development of epidermal melanocytes and enteric neurons

Amy Greenstein Baynash, Kiminori Hosoda, Adel Giaid et al. · Cell · 1994 · 957 citations

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