Total synthesis of the proposed structure of Dolastatin 15

Protection of hydroxyl groups as tert-butyldimethylsilyl derivatives

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Stereospecific synthesis of N-protected statine and its analogues via chiral tetramic acid

Patrick Jouin, Bertrand Castro, Dino Nisato · Journal of the Chemical Society Perkin Transactions 1 · 1987 · 189 citations

Natural Sciences, Chemistry, Medicinal Chemistry +13

Oxybenzotriazole free peptide coupling reagents for N-methylated amino acids

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