Biochemical and pharmacological properties of SR 49059, a new, potent, nonpeptide antagonist of rat and human vasopressin V1a receptors.

C. Serradeil‐Le Gal, Jean Wagnon, Corinne Garcia, +7

Journal of Clinical Investigation

Avp V2ImmunologyPharmacotherapyExperimental PharmacologyInflammation +16

Characterization of SR 121463A, a highly potent and selective, orally active vasopressin V2 receptor antagonist.

C. Serradeil‐Le Gal, C Lacour, G Valette, +17

Journal of Clinical Investigation

Molecular PharmacologySelective AffinityArginine VasopressinSr 121463AFunctional Selectivity +12

Characterization of (2 S,4 R)-1-[5-Chloro-1-[(2,4-dimethoxyphenyl)sulfonyl]-3-(2-methoxy-phenyl)-2-oxo-2,3-dihydro-1 H-indol-3-yl]-4-hydroxy-N,N-dimethyl-2-pyrrolidine carboxamide (SSR149415), a Selective and Orally Active Vasopressin V1b Receptor Antagonist

Claudine Serradeil‐Le Gal, Jean Wagnon, Jacques Simiand, +12

Journal of Pharmacology and Experimental Therapeutics

Stereospecific synthesis of N-protected statine and its analogues via chiral tetramic acid

Patrick Jouin, Bertrand Castro, Dino Nisato

Journal of the Chemical Society Perkin Transactions 1

Enantioselective SynthesisEngineeringStereospecific SynthesisMedicineN-protected Statine +11

A novel class of calcium-entry blockers: the 1-[[4-(aminoalkoxy)phenyl]sulfonyl]indolizines

J. Gubin, J. Lucchetti, Jean Mahaux, +5

Journal of Medicinal Chemistry

Electrophysiologic Characterization of Dronedarone in Guinea Pig Ventricular Cells

Patrick Gautier, Eric Guillemare, Aline Marion, +3

Journal of Cardiovascular Pharmacology

Cardiac MuscleHeart FailureAp AmplitudeElectrophysiologic CharacterizationCellular Physiology +14

Electrophysiological effects of dronedarone (SR 33589), a noniodinated amiodarone derivative in the canine heart: comparison with amiodarone

András Varró, J. Takács, Miklós Németh, +11

British Journal of Pharmacology

A new series of imidazolones: highly specific and potent nonpeptide AT1 angiotensin II receptor antagonists

C. BERNHART, Pierre Perreaut, B. Ferrari, +15

Journal of Medicinal Chemistry

Central Imidazole NucleusHealth SciencesImidazole SeriesFunctional SelectivityMedicine +10

Angiotensin AT1 Receptor Antagonist Irbesartan Decreases Lesion Size, Chemokine Expression, and Macrophage Accumulation in Apolipoprotein E-Deficient Mice

Frédérique Dol, Geneviève Martin, Bart Staels, +7

Journal of Cardiovascular Pharmacology

Vascular DiseaseImmunologyHyperlipidemiaPharmacotherapyInflammation +20

Inhibitory Effects of Dronedarone on Muscarinic K+ Current in Guinea Pig Atrial Cells

Eric Guillemare, Aline Marion, Dino Nisato, +1

Journal of Cardiovascular Pharmacology

Molecular PharmacologyCardiac MuscleInhibitory EffectsMedicinePhysiology +10