Concepedia

Structure–activity relationship study of thiosemicarbazones on an African trypanosome: Trypanosoma brucei brucei

Houssou Raymond Fatondji, Salomé Kpoviessi, Fernand Gbaguidi, Joanne Bero, Véronique Hannaert, Joëlle Quetin‐Leclercq, Jacques H. Poupaert, Mansourou Moudachirou, Georges C. Accrombessi

Medicinal Chemistry Research · 2012 · 45 citations · 24 references

DOI

Concepts

References

24

Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings

Christopher A. Lipinski, Franco Lombardo, Beryl W. Dominy et al. · Advanced Drug Delivery Reviews · 1997 · 11.2K citations

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The Alamar Blue® assay to determine drug sensitivity of African trypanosomes (T.b. rhodesiense and T.b. gambiense) in vitro

Barbara Räz, M Iten, Yvonne Grether-Bühler et al. · Acta Tropica · 1997 · 691 citations

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Cultivation in a semi‐defined medium of animal infective forms of Trypanosoma brucei, T. equiperdum, T. evansi, T. rhodesiense and T. gambiense.

T. Baltz, D. Baltz, C. Giroud et al. · The EMBO Journal · 1985 · 564 citations · Full text

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Synthesis and Structure−Activity Relationship Study of Potent Trypanocidal Thio Semicarbazone Inhibitors of the Trypanosomal Cysteine Protease Cruzain

Xiaohui Du, Chun Guo, Elizabeth Hansell et al. · Journal of Medicinal Chemistry · 2002 · 383 citations · Full text

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Synthesis, Cytotoxicity, and Antitumor Activity of Copper(II) and Iron(II) Complexes of <sup>4</sup><i>N</i>-Azabicyclo[3.2.2]nonane Thiosemicarbazones Derived from Acyl Diazines

Johnny Easmon, Gerhard Pürstinger, Gottfried Heinisch et al. · Journal of Medicinal Chemistry · 2001 · 255 citations

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