Rapid and automated tetrazolium-based colorimetric assay for the detection of anti-HIV compounds

Rudi Pauwels, Jan Balzarini, Masanori Baba, +5

Journal of Virological Methods

Medicinal ChemistryBioassay-guided IsolationTetrazolium-based Colorimetric AssayMedicineBioanalysis +10

High resolution structures of HIV-1 RT from four RT–inhibitor complexes

Jingshan Ren, Robert Esnouf, Elspeth F. Garman, +8

Nature Structural & Molecular Biology

BiochemistryNatural SciencesHuman RetrovirusHiv-1 RtAntiviral Drug Development +6

Discovery of 2,3-diaryl-1,3-thiazolidin-4-ones as potent anti-HIV-1 agents

Maria Letizia Barreca, Alba Chimirri, Laura De Luca, +8

Bioorganic & Medicinal Chemistry Letters

Medicinal ChemistryMedicineAntiviral Drug DevelopmentHivPharmacology +3

Carbodiimide mediated synthesis of 4-thiazolidinones by one-pot three-component condensation

Tumul Srivastava, W. Haq, S. B. Katti

Tetrahedron

Organic ChemistryOne-pot Three-component CondensationSynthetic ChemistryChemistry

Design, Synthesis, Structure−Activity Relationships, and Molecular Modeling Studies of 2,3-Diaryl-1,3-thiazolidin-4-ones as Potent Anti-HIV Agents

Maria Letizia Barreca, Jan Balzarini, Alba Chimirri, +9

Journal of Medicinal Chemistry

Combinatorial ChemistryBioorganic ChemistryChemistryPharmaceutical ChemistryMedicinal Chemistry +15

CP‐MLR/PLS Directed Structure‐Activity Modeling of the HIV‐1 RT Inhibitory Activity of 2,3‐Diaryl‐1,3‐thiazolidin‐4‐ones

Yenamandra S. Prabhakar, V. Raja Solomon, Ravindra K. Rawal, +2

QSAR & Combinatorial Science

Drug TargetPls ModelsPartial Least SquaresPharmaceutical ChemistryMolecular Pharmacology +15

A Combinatorial Approach to the Variable Selection in Multiple Linear Regression: Analysis of Selwood <i>et al.</i> Data Set – A Case Study

Yenamandra S. Prabhakar

QSAR & Combinatorial Science

EngineeringFeature SelectionRegression AnalysisVariable SelectionData Science +18

An expeditious synthesis of thiazolidinones and tetathiazanones

Ravindra K. Rawal, Tumul Srivastava, W. Haq, +1

Journal of Chemical Research

Combinatorial ChemistryRoom TemperatureBiochemistryNatural SciencesOrganic Chemistry +6

Topological Descriptors in Modeling the HIV Inhibitory Activity of 2-Aryl-3- pyridyl-thiazolidin-4-ones

Yenamandra S. Prabhakar, Ravindra K. Rawal, Manish Gupta, +2

Combinatorial Chemistry & High Throughput Screening

Topological DescriptorsDrug Target2-Aryl-3- Pyridyl-thiazolidin-4-onesMolecular BiologyAutocorrelation Descriptors +16

Synthesis and QSAR Studies on Thiazolidinones as Anti-HIV Agents

Ravindra K. Rawal, V. Raja Solomon, Yenamandra S. Prabhakar, +2

Combinatorial Chemistry & High Throughput Screening