Concepedia

Design, synthesis, and pharmacological evaluation of N-bicyclo-5-chloro-1H-indole-2-carboxamide derivatives as potent glycogen phosphorylase inhibitors

Kenichi Onda, Ryota Shiraki, Takashi Ogiyama, Kazuhiro Momose, Naoko Katayama, Masaya Orita, Tomohiko Yamaguchi, Masako Furutani, Noritaka Hamada, Makoto Takeuchi,

Bioorganic & Medicinal Chemistry · 2008 · 14 citations · 16 references

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16

Diphenylphosphoryl azide. New convenient reagent for a modified Curtius reaction and for peptide synthesis

Takayuki Shioiri, Kunihiro Ninomiya, Shun‐ichi Yamada · Journal of the American Chemical Society · 1972 · 938 citations

, , +6

An Efficient palladium-catalysed reaction of vinyl and aryl halides or triflates with terminal alkynes

Mouâd Alami, Fabiola Ferri, G. LINSTRUMELLE · Tetrahedron Letters · 1993 · 342 citations

, , +10

A new allosteric site in glycogen phosphorylase b as a target for drug interactions

Nikos G. Oikonomakos, Katerina E. Tsitsanou, Nikos G. Gavalas et al. · Structure · 2000 · 132 citations · Full text

, , +16

Flavopiridol Inhibits Glycogen Phosphorylase by Binding at the Inhibitor Site

Nikos G. Oikonomakos, Joachim Schnier, S.E. Zographos et al. · Journal of Biological Chemistry · 2000 · 125 citations · Full text

, , +11

Synergistic regulation of phosphorylase a by glucose and caffeine.

Peter J. Kasvinsky, Shirley Shechosky, Robert J. Fletterick · Journal of Biological Chemistry · 1978 · 112 citations · Full text

, , +15