Concepedia

Discovery and gram-scale synthesis of BMS-593214, a potent, selective FVIIa inhibitor

E. Scott Priestley, Indawati De Lucca, Jinglan Zhou, Jiacheng Zhou, Eddine Saiah, Robert V. Stanton, Leslie A. Robinson, Joseph M. Luettgen, Anzhi Wei, Xiao Wen,

Bioorganic & Medicinal Chemistry Letters · 2013 · 27 citations · 11 references

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11

Lanthanide Triflate Catalyzed Imino Diels-Alder Reactions; Convenient Syntheses of Pyridine and Quinoline Derivatives

Shū Kobayashi, Haruro Ishitani, Satoshi Nagayama · Synthesis · 1995 · 226 citations

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A New Methodology for Combinatorial Synthesis. Preparation of Diverse Quinoline Derivatives Using a Novel Polymer-Supported Scandium Catalyst

Shū Kobayashi, Satoshi Nagayama · Journal of the American Chemical Society · 1996 · 176 citations

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Antithrombotic Effects of Recombinant Human, Active Site–Blocked Factor VIIa in a Rabbit Model of Recurrent Arterial Thrombosis

Paolo Golino, Massimo Ragni, Plinio Cirillo et al. · Circulation Research · 1998 · 77 citations · Full text

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Pharmacological Interruption of Acute Thrombus Formation with Minimal Hemorrhagic Complications by a Small Molecule Tissue Factor/Factor VIIa Inhibitor: Comparison to Factor Xa and Thrombin Inhibition in a Nonhuman Primate Thrombosis Model

Osman D. Suleymanov, James A. Szalony, Anita K. Salyers et al. · Journal of Pharmacology and Experimental Therapeutics · 2003 · 64 citations

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A Selective, Slow Binding Inhibitor of Factor VIIa Binds to a Nonstandard Active Site Conformation and Attenuates Thrombus Formation in Vivo

Alan G. Olivero, Charles Eigenbrot, Richard Goldsmith et al. · Journal of Biological Chemistry · 2005 · 41 citations · Full text

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