Reaction of N -alkyl azetidines with triphosgene

Synthesis and Profiling of a Diverse Collection of Azetidine-Based Scaffolds for the Development of CNS-Focused Lead-like Libraries

Jason T. Lowe, Maurice D. Lee, Lakshmi B. Akella et al. · The Journal of Organic Chemistry · 2012 · 137 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +16

Azetidines: New Tools for the Synthesis of Nitrogen Heterocycles

François Couty, Gwilherm Evano · Synlett · 2009 · 117 citations

Natural Sciences, Chemistry, Medicinal Chemistry +12

Discovery and Optimization of an Azetidine Chemical Series As a Free Fatty Acid Receptor 2 (FFA2) Antagonist: From Hit to Clinic

Mathieu Pizzonero, Sonia Dupont, Marielle Babel et al. · Journal of Medicinal Chemistry · 2014 · 110 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

Enantioselective Syntheses of Morpholines and Their Homologues via S_N2-Type Ring Opening of Aziridines and Azetidines with Haloalcohols

Manas K. Ghorai, Dipti Shukla, Kalpataru Das · The Journal of Organic Chemistry · 2009 · 101 citations

Natural Sciences, Chemistry, Medicinal Chemistry +13

Preparation and Synthetic Applications of Azetidines

F. G. West, Tina M. Bott · Heterocycles · 2011 · 93 citations · Full text

Natural Sciences, Chemistry, Medicinal Chemistry +15