Mathieu Pizzonero

Discovery and Optimization of an Azetidine Chemical Series As a Free Fatty Acid Receptor 2 (FFA2) Antagonist: From Hit to Clinic

Mathieu Pizzonero, Sonia Dupont, Marielle Babel et al. · Journal of Medicinal Chemistry · 2014 · 107 citations · Full text

Inflammation, From Hit, Medicinal Chemistry +15

The syntheses of rac-inthomycin A, (+)-inthomycin B and (+)-inthomycin C using a unified synthetic approach

Michael R. Webb, Matthew S. Addie, Catherine M. Crawforth et al. · Tetrahedron · 2008 · 56 citations

Bioorganic Chemistry, Engineering, Biochemistry +10

Identification of GLPG/ABBV-2737, a Novel Class of Corrector, Which Exerts Functional Synergy With Other CFTR Modulators

Gert De Wilde, Maarten Gees, Sara Musch et al. · Frontiers in Pharmacology · 2019 · 39 citations · Full text

Protein Secretion, Other Cftr Modulators, Molecular Physiology +11

X-Ray Crystal Structures of Potent Receptor Ligands: Etonitazene, cis-(+)-3-Methylfentanyl, Etorphine, Diprenorphine, and Buprenorphine

Mathieu Pizzonero, J.L. Flippen-Anderson, Clifford George et al. · Heterocycles · 1994 · 21 citations · Full text

X-ray Crystallography, Drug Target, Potent Receptor +18

Discovery of Pyridones As Oral AMPK Direct Activators

Olivier Mirguet, Stéphane Sautet, Catherine-Anne Clément et al. · ACS Medicinal Chemistry Letters · 2013 · 14 citations · Full text

Medicinal Chemistry, Pharmaceutical Science, Biochemistry +11