Concepedia

Cannabinoid Partial Agonists

Cannabinoid Partial Agonist is a pharmacological agent that binds to and activates cannabinoid receptors with submaximal efficacy relative to full agonists, thereby producing a diminished downstream signaling response despite complete receptor occupancy.

116

Publications

6.6K

Citations

520

Authors

185

Institutions

Publications per year

2017–2026

19

Variants

Cannabinoid Partial Agonist

Parents

Publications

116

Anandamide, an endogenous cannabinoid, inhibits calcium currents as a partial agonist in N18 neuroblastoma cells.

Ken Mackie, William A. Devane, Bertil Hille · Molecular Pharmacology · 1993 · 362 citations

, , +16

The Activity of Anandamide at Vanilloid VR1 Receptors Requires Facilitated Transport across the Cell Membrane and Is Limited by Intracellular Metabolism

Luciano De Petrocellis, Tiziana Bisogno, Mauro Maccarrone et al. · Journal of Biological Chemistry · 2001 · 352 citations · Full text

, , +15

Evidence That the Cannabinoid CB1 Receptor Is a 2-Arachidonoylglycerol Receptor

Takayuki Sugiura, Tomoko Kodaka, Shinji Nakane et al. · Journal of Biological Chemistry · 1999 · 313 citations · Full text

, , +14

Rapid assessment of a novel series of selective CB2 agonists using parallel synthesis protocols: A Lipophilic Efficiency (LipE) analysis

Thomas Ryckmans, Martin P. Edwards, Val A. Horne et al. · Bioorganic & Medicinal Chemistry Letters · 2009 · 269 citations · Full text

, , +17

Conditioned place preference induced by Δ9-tetrahydrocannabinol: comparison with cocaine, morphine, and food reward

Marino Lepore, Stanislav R. Vorel, Joyce H. Lowinson et al. · Life Sciences · 1995 · 239 citations

, , +14

1–5 of 116

Authors

520

  1. BR
    Billy R. Martin

    Virginia Commonwealth University Medical Center, United States

    13 publications · 547 citations

    13

    h-index

  2. RG
    Roger G. Pertwee

    University of Aberdeen, United Kingdom

    9 publications · 540 citations

    9

    h-index

  3. JL
    Jenny L. Wiley

    RTI International, United States

    7 publications · 252 citations

    7

    h-index

  4. AM
    Alexandros Makriyannis

    Northeastern University, United States

    6 publications · 301 citations

    6

    h-index

  5. RK
    Raj K. Razdan

    Organix (United States), United States

    6 publications · 212 citations

    6

    h-index

1–5 of 520

Institutions

185

  1. Virginia Commonwealth University Medical Center

    Richmond, United States

    11 h-index

    30 publications

    1.2K citations

  2. University of Aberdeen

    Aberdeen, United Kingdom

    8 h-index

    22 publications

    1.6K citations

  3. University of Connecticut

    Storrs, United States

    5 h-index

    16 publications

    744 citations

  4. Virginia Commonwealth University

    Richmond, United States

    4 h-index

    12 publications

    597 citations

  5. Northeastern University

    Boston, United States

    4 h-index

    18 publications

    716 citations

  6. Universidad Complutense de Madrid

    Madrid, Spain

    4 h-index

    22 publications

    1.5K citations

  7. Clemson University

    Clemson, United States

    4 h-index

    10 publications

    427 citations

  8. National Institutes of Health

    Bethesda, United States

    3 h-index

    11 publications

    371 citations

1–8 of 185

Venues

  1. Journal of Medicinal Chemistry

    10 publications · 504 citations

    10

    h-index

  2. Behavioural Pharmacology

    11 publications · 501 citations

    10

    h-index

  3. British Journal of Pharmacology

    BJP · 10 publications · 539 citations

    10

    h-index

  4. 7

    h-index

  5. European Journal of Pharmacology

    EJP · 6 publications · 137 citations

    6

    h-index

1–5