Lee R. Roberts

A road map to evaluate the proteome-wide selectivity of covalent kinase inhibitors

Bryan Lanning, Landon R. Whitby, Melissa M. Dix et al. · Nature Chemical Biology · 2014 · 356 citations · Full text

Molecular Docking, Drug Target, Biochemistry +10

Gut microbial β-glucuronidases reactivate estrogens as components of the estrobolome that reactivate estrogens

Samantha M. Ervin, Hao Li, Lauren Lim et al. · Journal of Biological Chemistry · 2019 · 340 citations · Full text

Biosynthesis, Biochemistry, Endocrine Research +15

Design and Structure of Stapled Peptides Binding to Estrogen Receptors

Chris Phillips, Lee R. Roberts, Markus Schade et al. · Journal of the American Chemical Society · 2011 · 248 citations

Biochemistry, Stapled Peptides, Protein Folding +15

Rational Targeting of Active-Site Tyrosine Residues Using Sulfonyl Fluoride Probes

Erik C. Hett, Hua Xu, Kieran F. Geoghegan et al. · ACS Chemical Biology · 2015 · 191 citations

Molecular Pharmacology, Drug Target, Biochemistry +15

( <i>R</i> )-PFI-2 is a potent and selective inhibitor of SETD7 methyltransferase activity in cells

Dalia Baršytė-Lovejoy, Fengling Li, Menno J. Oudhoff et al. · Proceedings of the National Academy of Sciences · 2014 · 188 citations · Full text