<i>S</i>-Acyl-2-thioethyl Phosphoramidate Diester Derivatives as Mononucleotide Prodrugs

David Egron, Jean‐Louis Imbach, Gilles Gosselin, +2

Journal of Medicinal Chemistry

Bioorganic ChemistryNew SeriesAntiviral DrugChemical BiologyPharmaceutical Chemistry +14

New bis(SATE) prodrug of AZT 5′‐monophosphate: In vitro anti‐HIV activity, stability, and potential oral absorption

Manijeh Shafiee, S. Deferme, Anne‐Laure Villard, +11

Journal of Pharmaceutical Sciences

Medicinal ChemistryPharmaceutical ScienceMedicineAntiviral Drug DevelopmentNew Bis +10

Analysis of neutral lipids from microalgae by HPLC-ELSD and APCI-MS/MS

Florentin Donot, Guillaume Cazals, Ziya Günata, +5

Journal of Chromatography B

Lipid AnalysisEngineeringBiochemistryBioanalysisMass Spectrometry +7

Radical cyclization of highly functionalized precursors: stereocontrol of ring closure of acyclic 1-substituted-2,4-dihydroxylated hex-5-enyl radicals

Arlène Roland, Thierry Durand, David Egron, +2

Journal of the Chemical Society Perkin Transactions 1

DerivativesEngineeringNatural SciencesAll-syn PrecursorDiversity-oriented Synthesis +11

Identification of Noncompetitive Inhibitors of Cytosolic 5′-Nucleotidase II Using a Fragment-Based Approach

Zsuzsanna Márton, Rémi Guillon, Isabelle Krimm, +10

Journal of Medicinal Chemistry

Biolabile constructs for pronucleotide design

A.M. Jochum, Nathalie Schlienger, David Egron, +2

Journal of Organometallic Chemistry

Natural SciencesBiolabile ConstructsSynthetic BiologyMolecular BiologyDna Replication +6

Anti-HIV pronucleotides: Decomposition pathways and correlation with biological activities

David Egron, Isabelle Lefèbvre, Christian Périgaud, +5

Bioorganic & Medicinal Chemistry Letters

Anti-hiv PronucleotidesNatural SciencesHuman RetrovirusAntiviral ResponseMolecular Biology +5

Increase of the adenallene anti-HIV activity in cell culture using its bis(tBuSATE) phosphotriester derivative

David Egron, Christian Périgaud, Gilles Gosselin, +5

Bioorganic & Medicinal Chemistry Letters

Adenallene Anti-hiv ActivityBiochemistryMedicineAntiviral Drug DevelopmentCell Culture +5

Rational design of a new series of pronucleotide

Thierry Beltran, David Egron, Alain Pompon, +5

Bioorganic & Medicinal Chemistry Letters

Natural SciencesOligonucleotideDna ReplicationSynthetic BiologyMolecular Biology +3

Antiviral Activity and Intracellular Metabolism of Bis(tButylSATE) Phosphotriester of β-L-2′,3'Dideoxyadenosine, a Potent Inhibitor of HIV and HBV Replication

L Placidi, Achraf Al Faraj, AG Loi, +11

Antiviral chemistry & chemotherapy